Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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166
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180
of
65,077
results
166
Tocris Bioscience™ YKL 5-124
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective CDK7 inhibitor; induces cell cycle arrest
167
Tocris Bioscience™ BRD 0539
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Cell permeable and reversible Cas9 inhibitor
| Target | CRISPR Reagents |
|---|---|
| CAS | 1403838-79-8 |
| Purity | 0.98 |
| Chemical Name or Material | (3 aR,4 R,9 bR)-8-(2-Fluorophenyl)-2,3,3 A,4,5,9 b-hexahydro-1-[(4-methylphenyl)sulfonyl]-1 H-pyrrolo[3,2-c]quinoline-4-methanol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H25FN2O3S |
168
Tocris Bioscience™ Erlotinib Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent, reversible EGFR tyrosine kinase inhibitor
169
Tocris Bioscience™ Dooku 1
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Reversibly blocks Yoda1 activity; does not affect constitutive Piezo1 activity
| Target | Other Piezo Channel Compounds |
|---|---|
| CAS | 2253744-54-4 |
| Purity | 98% |
| Chemical Name or Material | 2-[(2,6-Dichlorobenzyl)thio)-5-(1 H-pyrrol-2-yl)-1,3,4-oxadiazole |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C13H9Cl2N3OS |
| Formula Weight | 326.2 |
170
Tocris Bioscience™ THAL SNS 032
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective Cdk9 Degrader (PROTAC™)
171
| CAS | 19685-09-7 |
|---|---|
| Molecular Formula | C20H16N2O5 |
172
Tocris Bioscience™ Carfilzomib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent irreversible proteasome inhibitor; active in vivo
| Target | Proteasome Inhibitors |
|---|---|
| CAS | 868540-17-4 |
| Purity | 0.98 |
| Chemical Name or Material | (αS)-α-[[2-(4-Morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-N-[(1 S)-3-methyl-1-[[(2 R)-2-methyl-2-oxiranyl]carbonyl]butyl]-L-phenylalaninamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C40H57N5O7 |
173
Tocris Bioscience™ PF 04449913 maleate
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent Smo antagonist
| CAS | 2030410-25-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 1-((2R,4R)-2-(1H-Benzimidazol-2-yl)-1-methylpiperidin-4-yl)-3-(4-cyanophenyl)urea maleate salt |
| Recommended Storage | Store at -20°C |
| Synonym | glasdegib, PF-913 |
| Molecular Formula | C21H22N6O.C4H4O4 |
174
Tocris Bioscience™ BDY FL VH032
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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High-affinity VHL fluorescent probe for TR-FRET and FP assays
175
Tocris Bioscience™ Lac-Phe
Metabolite generated by cytosol nonspecific dipeptidase (CNDP2) during intense exercise
| Target | DNA, RNA and Protein Synthesis Compounds |
|---|---|
| CAS | 183241-73-8 |
| Purity | 0.95 |
| Chemical Name or Material | N-[(2S)-2-Hydroxy-1-oxopropyl]-L-phenylalanine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C12H15NO4 |
176
Tocris Bioscience™ uPSEM 792 hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Highly potent PSAM4-GlyR and PSAM4-5-HT3 chimeric ion channel agonist; brain-penetrant
| Target | Pharmacologically Selective Effector Molecules/PSEM |
|---|---|
| CAS | 2341841-08-3 |
| Purity | 98% |
| Chemical Name or Material | 1-Methyl-7,8,9,10-tetrahydro-1 H-6,10-methanoazepino[4,5-g]quinoxalin-2(6 H)-one hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C14H15N3O.HCl |
| Formula Weight | 277.75 |
177
Tocris Bioscience™ Veliparib dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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High affinity PARP-1 and -2 inhibitor; orally bioavailable
178
Tocris Bioscience™ CG 858-Neg
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Negative control for CG 858 (Cat. No. 7427)
179
Tocris Bioscience™ CG 428
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent tropomyosin receptor kinase (TRK) degrader
180
Tocris Bioscience™ Phalloidin-FITC
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Green fluorescent cytoskeleton stain